cas 1809278-35-0 Tianeptine ethyl ester sulfate cas 66981-77-9

drum

What Is Tianeptine?

Stablon/Coaxil, also known as Tianeptine is a pharmaceutical-grade compound that is often used for the treatment of clinical depression. It is also sometimes used to help mitigate the symptoms of asthma and irritable bowel syndrome.

At large doses, tianeptine is known to produce opioid-like recreational effects, such as stimulation and sedation, motivation, and euphoria. In terms of classification, tianeptine is a tricyclic antidepressant.

However, it’s effects and pharmacology vary from a traditional anxiolytic and antidepressant. Primarily in the fact that it does not act immediately through regulation of monoaminergic neurotransmitters, such as noradrenaline, dopamine, and serotonin. But rather acts upon glutamatergic and glutamate mechanisms, causing the brain to adapt to depression and stress.

In a clinical setting, it is suggested that tianeptine is just as effective as typical antidepressants, such as amitryptiline and fluoxetine. In addition to that, it seems to exhibit fewer side effects and associated complications.

Not to mention, tianeptine has a strong anxiolytic profile, showing lots of promise in treating panic disorders. Tianeptine also has some effect on cognition and neuroprotective properties of the brain. Considering all of the above, tianeptine is a popular nootropic